Publications

Publications

We have published in the following prestigious journals:

  • Anal. Chem.
  • Journal of Chromatography
  • Electrophoresis
  • Org. Chem.
  • Phys. Org. Chem
  • Chem. Crystallography
  • Tetrahedron
  • Indian J. Chem.
  • Clinical Pharmacokinetics
  • Clinical Pharmacology and Therapeutics
  • Cancer Research
  • National Institutes of Health
  • American Chemical Society
  • Acta Pharmaceutica Sinica
  • Annual Meeting of American Association for Cancer Research (AACR)
  • Associations of Officials in Analytical Chemistry (AOAC)
  • Chinese Chemical Letters
  • Chinese Pharmaceutical Journal
  • Chinese Traditional and Herbal Drugs
  • Journal of Pharmaceutical and Biomedical Analysis (JPBA)
  • Encyclopedia of Agrochemicals
  • Fitoterapia
  • Journal of Natural Products
  • Natural Product Research
  • Planta Medica
  • Journal of Pesticide Science
  • Journal of Agricultural and Food Chemistry
  • Nuclear Instruments and Methods in Physics Research
  • Environmental Science and Technology
  • R. Bartnik, Macromol. Symp.

Publications:

  • Safarpour, H., Connolly P., Tong X.J., Bielawski, M., and Wilcox E. "Overcoming extractability hurdles of a 14C-labled taxane analogue-milataxel and its metabolite from xenograft mouse tumor and brain tissues." Journal of Pharmaceutical and Biomedical Analysis (49)3, 774-9 (2009).
  • Safarpour, H., Tong, X., Bielawski, M., Holton, R., and Wilcox, H. "Concentration of Milataxel (MAC-321, TL-139) and its major metabolite (M-10) in xenograft tumors from mice dosed orally and intravenously." Proceedings of 97th AACR, April 2006.
  • Gu, J.Q., Tong, X.J., Ding, Y., Fang, Q.C. "Application of high-speed countercurrent chromatography to the separation of taxol and cephalomannine." Fitoterapia 65(2), 149-52 (1994).
  • Hall, A.M., Tong, X.J., Chang, C. "Taxoids from Taxus x media 'Dark Green Spreader.'" Natural Product Research (10)3, 165-72 (1997).
  • Harris, N., Griffin, M., Turner, K., Safarpour, H., Wilcox, E., Boddy, A. "Metabolism of the oral taxane TL310 in vitro and in a Phase I study." Proceedings of 100th Annual Meeting of American Association for Cancer Research (AACR), April 2009.
  • Holton, R., Metts, L., Abramowitz, R., Arrington, H., Edler, M., Wilcox, E., Williams, A., Zorlo, D. "Preclinical evaluation of TL-1892, a novel orally active taxane with superior in vitro and in vivo efficacy in paclitaxel and docetaxel resistant models." AACR abstract #723
  • Holton, R., Metts, L., Abramowitz, R., Arrington, H., Edler, M., Wilcox, E., Williams, A., Zorlo, D. "TL-1836, A new orally active taxane with curative antitumor activity against human tumor xenografts." AACR abstract #1401.
  • Longley, R.E., Clement, C., Metts, L., Holton, R. "In vivo efficacy of TL-310: A new, orally active taxane analog." AACR abstract #7363. 2006.
  • Ohba, K., Minoura, M., Picard, G., and Safarpour, H. "Method for the determination of imazamox and its two hydroxy and glucose conjugate metabolites in adzuki beans by capillary electrophoresis." Journal of Pesticide Science, 22(4), 277-81 (1997).
  • Safarpour, H., Asiaie R. "Capillary Electrophoresis (CE)-Its Application to Pesticide Analysis." Encyclopedia of Agrochemicals, 2001, John Weily & Sons.
  • Safarpour, H., Asiaie R. "Determination of Glyphosate as cross-contaminant in a commercial herbicide by capillary electrophoresis-electrospray ionization-mass spectrometry." Electrophoresis 26(7-8), 1562-6 (2005).
  • Safarpour, H., Asiaie R. "Quantitaive analysis of imazamox herbicide in environmental water samples by capillary electrophoresis electrospray ionization mass spectrometry." Journal of Chromatography A, 1036(2), 217-222 (2004).
  • Tong, X.J., Fang, W.S., Fang, Q.C. "Studies on the chemical constituents of Taxus cuspidata." Chinese Chemical Letters 4, 887 (1993).
  • Tong, X.J., Fang, W.S., Fang, Q.C. "Studies on chemical constituents of Taxus cuspidata." Acta Pharmaceutica Sinica 29, 55 (1994).
  • Tong, X.J., Fang, W.S., Zhou, J.Y., He, C.H., Chen, W.M., Fang, Q.C. "Three new taxane diterpenoids from needles and stems of Taxus cuspidata." Journal of Natural Products 58(2), 233-38 (1995).
  • Tong, X.J., Liu, Y.C., Chang, C.J. "Taxanes from Taxus x media Hicksii." Natural Product Research 6(3), 197-202 (1995).
  • Tong, X.J., Wang, H.B., Fang, Q.C. "Studies on the alkaloids from the fermentation product of Claviceps paspali." Chinese Traditional and Herbal Drugs 23, 103 (1992).
  • Tong, X.J., Zhou, J.Y., Fang, Q.C. "Chemical constituents of Pygeum topengii." Chinese Pharmaceutical Journal 28(3), 133 (1993).
  • Zhou, J.Y., Chen, B.Z., Tong, X.J., Fang, Q.C. "Chemical study on the alkaloids of Chelidonium majus L." Chinese Traditional and Herbal Drugs 20, 2 (1989).
  • Zhou, J.Y., Tong, X.J., Fang, Q.C. "Chemical studies on the alkaloids of Corydalis hsuchowensis." Planta Medica 57(2), 156-8 (1991).
  • Ingle N, Buzdar AU, Schaid DJ, Goetz MP, Batzler A, Robson ME, Northfelt DW, Olson JE, Perez EA, Desta Z, Weintraub RA, Williard CV, Flockhart DA, Weinshilboum RM. Variation in Anastrozole Metabolism and Pharmacodynamics in Women with Early Breast Cancer, Cancer Research, 70(8), 3024-3033 (2010)
  • Weintraub RA, Ameer B, Johnson JV, Yost RA. Trace Determination of Naringenin and Hesperitin by Tandem Mass Spectrometry, Journal of Agricultural and Food Chemistry, 43, 1966-1968 (1995)
  • Ameer B, Weintraub RA, Johnson JV, Yost RA, Rouseff RL. Flavanone Absorption after Naringin, Hesperidin and Citrus Administration, Clinical Pharmacology and Therapeutics, 60, 34-40, (1996)*
  • Ameer B, Weintraub RA. Drug Interactions with Grapefruit Juice, Clinical Pharmacokinetics, 33(2), 103-121 (1997)*
  • Jibaly M, Chrusch P, Hilgenberg G, Majewski S, Wojcik R, Weintraub R, Sauli, F. Some Results on the Ageing of Wire Chambers with Dimethyl Ether, Nuclear Instruments and Methods in Physics Research Section A, 273(1), 161-171 (1988)
  • Moye HA, Weintraub RA. “Correspondence: Comments on Reaction Products and Rates of Disappearance of Simple Bromoalkanes, 1,2-dibromopropane and 1,2-dibromoethane in Water,” Environmental Science and Technology; 2, 231 (1987)
  • Moye, HA, Weintraub, RA, Jex, GW, "Modes of Ethylene Dibromide Degradation," Final report to Florida Department of Environmental Regulation, Gainesville, Florida, University of Florida Pesticide Research Laboratory (1987)
  • Weintraub RA, Jex GW, Moye HA. “Chemical and Microbial Degradation of 1,2-Dibromoethane (EDB) in Florida Groundwaters, Soils and Sludge,” in Evaluation of Pesticides in Ground Water, American Chemical Society Sympos. Series; 315, Chap.15, 294-310, Honeycutt R, Garner W, Nigg H Eds. (1986)
  • Deyrup CL, Chang S, Weintraub RA, Moye HA. Simultaneous Esterification and Acylation of Pesticides for Analysis by Gas Chromatography. 1. Derivatization of Glyphosate and (Aminomethyl)-Phosphonic Acid with Fluorinated Alcohols-Perfluorinated Anhydrides, Journal of Agricultural and Food Chemistry; 33, 944-948 (1985)
  • Synthesis and Inclusion complexation studies of a Novel and selective receptor for 1,4-disubstituted benzene and 4,4’-disubstittuted biphenol, Macias A. T., Kumar. K.A., Marchand A.P., Evanseck J.D., J.Org. Chem., 2000, 65, 2083.
  • Convenient Deprotective Acylative Dealkylation of Tertiary Amines, T. Axenrod, R. Dai, K.K. Das, P.R. Dave, R. Duddu, X.P. Guan, K.A. Kumar, J. Sun, N. Trivedi, J.Org. Chem., 2000, 65, 1207.
  • Selective extraction of Lead(II) into Chloroform by lipophilic dibenzopolyether dicarboxylic acids possessing different spacer units, T. Hayashita, T. Higuchi, T. Fujimoto, A.P. Marchand, K.A. Kumar, N. Elkarim, H. Hwang, R.A. Bartsch, Talanta,, 2000, 52, 385.
  • Evaluation of Binding Selectivities of Caged Crown Ligands Towards Heavy Metals by Electrospray Ionization/Quadrupole Ion Trap Mass Spectrometry, Blair S.M,. Brodbeldt J.S,. Marchand A.P,. Kumar K.A,. Chong H.-S. Anal. Chem.,2000, 72, 2433.
  • Structure of Deaza Dimer of 4-methyl-3H-1,2,4-triazole-3,5(4H)-dione, S.G. Bott, A.P. Marchand, K.A. Kumar, D. Xing, J. Chem. Crystallogr., 1999, 29, 15.
  • Synthesis and structure of a bis(ethynyl)-substituted oxahexacyclic cage ether, S.G. Bott, A.P. Marchand, K. A. Kumar, J. Chem. Crystallogr., 1999, 29, 347.
  • New Adventures with Divalent carbon Intermediates, A.P. Marchand, D. Rajagopal, K.A. Kumar, R. Eckrich, K.C.V. Ramaniah, I.N.N. Namboothiri, S. Alihodzic, E.Z. Dong, R. Shukla, S.G. Bott, G. Mloston, A. Galindo, R. Bartnik, Macromol. Symp., 1998, 114, 95.
  • Synthesis and Alkali Metal Picrate Extraction Capabilities of a 4-Oxahexacyclo [5.4.1.02,6. 03,10.05,9.08,11]dodecane-derived Cryptand. A New Ionophore for selective Ion complexation, A.P. Marchand, S. Alihodzic, A.S. McKim, K. A. Kumar, K.M. Majerski, T. Sumanovac, S.G. Bott, Tetrahedron Lett., 1998, 39, 1861.
  • Synthesis and Alkali Metal Picrate Extraction Capabilities of Novel, Cage-Functionalized Diazacrown Ethers. Effects of Host Preorganization on Avidity and Selectivity Towards Alkali Metal Picrates in Solution, A.P. Marchand, A.S. McKim, K.A. Kumar, Tetrahedron, 1998, 54, 13421.
  • Intermolecular vs. Intramolecular Carbene Reactions of a Cage-Functionalized Cyclopentylcarbene, A.P. Marchand, K. A. Kumar, K. M. Majerski, J. Veljkovic, Tetrahedron, 1998, 54, 15105.
  • Crystal Structures of Three Substituted Pentacyclo[5.4.0.02,6.03,10.05,9]undecanes, S.G. Bott, A.P. Marchand, S. Alihodzic, K.A. Kumar, J. Chem. Crystallogr., 1998, 28, 251.
  • Inclusion Complexation of cyclobis(paraquat-p-phenylene) and Related Cyclophane Derivatives with Substituted Aromatics: Cooperative Non-Covalent Cavity and External Interactions, R. Castro, P.D. Davidov, K. A. Kumar, A.P. Marchand, J.D. Evanseck, A.E. Kaifer, J. Phys. Org. Chem, 1997, 10, 369.
  • Synthesis and Alkali Metal Picrate Extraction Capabilities of Novel Cage-Functionalized 17-Crown-5 and 17-Crown-6 Ethers, A.P. Marchand, K.A. Kumar, A.S. McKim, K.M. Majerski, G. Kragol, Tetrahedron, 1997, 53, 3467.
  • Acid and Base Promoted Rearrangments of Hexacyclo[11.2.02,12.05,10.05,15.010,14] hexadeca-6,8-diene-4,11-dione, A.P.Marchand, H. Soon, R. Shukla, G.V. M. Sharma, K.A. Kumar, U.R. Zope, S.G. Bott, Tetrahedron , 1996, 52, 13531.
  • Reaction of Vinylmagnesium Bromide with Hexacyclo[10.2.1.04,9.04,14.09,13] pentadeca-5,7-diene-3,10-dione: Transannular Hemiketal Formation, S.G. Bott, A.P. Marchand, K.A. Kumar, J. Chem. Crystallogr. , 1996, 26, 429.
  • Tetracyclo[6.3.0.04,11.05,9]undeca-2,7-dione, S.G. Bott, D. Rajagopal, K. A. Kumar, A.P. Marchand, J. Chem. Crystallogr., 1996, 26, 425.
  • Structure of 1-(2’-Tosyloxyethoxy)-8-tosyloxy-9,10-anthraquinone, S.G. Bott, A.P. Marchand, K. A. Kumar, J. Chem. Crystallogr., 1996, 26, 677.
  • Generation and Trapping of a Caged Cyclopentylidenecarbene, A. P. Marchand, K. A. Kumar,
    D. Rajagopal, R. Eckrich, S. G. Bott, Tetrahedron Lett., 1996, 37, 467.
  • Thermodynamic vs. Kinetic Control in the Diels-Alder Cycloaddition of Cyclo-pentadiene to 2,3-Dicyano-p-Benzoquinone, A. P. Marchand, K. A. Kumar, S. G. Bott, J. Chem. Crystallogr., 1996, 26, 281.
  • Synthesis, Characterization and Crystal Density Modeling of Polycarbocyclic Oxiranes, A.P. Marchand, D. Vidyanand, Z. Liu, K.A. Kumar, F. Zaragoza, S.G. Bott, W.H. Watson, R.P. Kashyap, H.L. Ammon, Z. Du, Tetrahedron, 1996, 52, 9703.
  • A Novel Reduction(Zn/AcOH) of DDHQ Esters- A new Route to Tropone Synthesis, T.R. Kasturi, P.V.P. Palle, J.A. Sattigeri, K. A. Kumar, Tetrahedron, 1996, 52, 1707.
    Syntheses of Bis- and Tetra-crowned Clefts and Studies of their Selectivities in Metal Ion complexation, R.A. Bartsch, M. Eley, A.P. Marchand, R. Shukla, K.A. Kumar, G. M. Reddy, Tetrahedron, 1996, 52, 8979.
  • A new Synthesis of Dibenzo[aj]xanthene derivatives., T.R. Kasturi and K. A. Kumar, Indian J. Chem., 1995, 34B, 6.
  • Synthesis and Thermal rearrangment of Pentacyclo[6.5.0.04,12.05,10.09,13]trideca-2,6-diene, A. P. Marchand, D. Rajapaksa, V. Vidyasagar, R. Eckrich, K. A. Kumar, Tetrahedron, 1995, 51, 11937.
  • Nucleophilic Additions of Primary and Secondary Amines to Pentacyclo [6.5.0. 04,12.05,10.09,13] undeca-8,11-dione, S. G. Bott, A.P. Marchand, K. A. Kumar, D. Vidyanand, D. Xing, W. H. Watson, R. Kashyap, R. A. Sachleben, J. Chem. Crystallogr, 1995, 25, 633.
  • A Novel Stereoselective Synthesis of (Z)-3-Iodo-3-alken-1-ones from 2-alkyn-1-ones. Fen-Tair Luo, K. A. Kumar, Li-Chen Hsieh and Ren-Tzong Wang, Tetrahedron Lett., 1994, 35, 2553.
  • Reaction of Spironaphthalenones with Hydroxylamine Hydrochloride Part III. A novel Mechanism for the formation of Products. Trapping of an Intermediate. T.R. Kasturi, K. A. Kumar, P.V.P.P.Charyulu, G.Sridevi, Tetrahedron, 1993, 49, 134.
  • Reaction of Spironaphthalenones with Hydroxylamine Hydrochloride Part II. Reaction of 1'-Substituted Spironaphthalenones -Structure of Products. T.R. Kasturi, K. A. Kumar and P.V.P.P. Charyulu, Tetrahedron, 1993, 49, 125.
  • Reaction of spironaphthalenones with Hydroxylamine Hydrochloride Part I. A reinvenstigation of the Mechanism. T.R.Kasturi, S.K. Jayaram, P.V.P.P. Charyulu, G.M. Reddy and K. A. Kumar, Tetrahedron, 1993, 49, 113.
  • Synthesis of (+)-1-t-butoxy-3a,6,7,7a-tetrahydro-7a-alkylindanes-New chiral synthons. T.R. Kasturi, R. Saibaba., K. A. Kumar and D.K. Banerjee, Indian J. Chem., 1990, 29B, 1083.

* Listed in the National Institutes of Health Bibliography (CBM99-04) on the Bioavailability of Nutrients and other Active Components of Dietary Supplements: http://www.nlm.nih.gov/archive/20040829/pubs/cbm/bioavailability.html